After release into the synaptic cleft, the neurotransmitter dopamine is actively taken up
by the cells via specific dopamine transporters. The drug cocaine interferes with this
process and is therefore called a reuptake inhibitor. The inhibition of the transporter at a
certain cocaine concentration is qualitatively represented in the following graph. Based
on this graph, which of the following describes the effect of cocaine on the kinetics of
dopamine reuptake by the transporter?
A.In the presence of cocaine, the maximal rate of transport (Vmax) is unaffected, but the
apparent affinity of the transporter for dopamine is reduced.
B.In the presence of cocaine, the maximal rate of transport (Vmax) is reduced, but the
apparent affinity of the transporter for dopamine is unaffected.
C.In the presence of cocaine, the maximal rate of transport (Vmax) is enhanced, but the
apparent affinity of the transporter for dopamine is unaffected.
D.In the presence of cocaine, both the maximal rate of transport (Vmax) and the
apparent affinity of the transporter for dopamine are enhanced.
E.In the presence of cocaine, both the maximal rate of transport (Vmax) and the
apparent affinity of the transporter for dopamine are unaffected, but the transporter is
nevertheless inhibited.
You grow neurons in culture in the presence or absence of nerve growth factor (NGF).
You perform this experiment using either wild-type neurons or neurons lacking
caspase-3, an effector protein required for programmed cell death by apoptosis in these
cells. After a day, you examine cell survival in the culture using a microscope. The
survival scores (percentage of cells surviving the treatment) are presented in the
following table. Which column (a or b) corresponds to the experiment in the presence
of NGF? Which row (1 or 2) corresponds to the experiment using wild-type cells?